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Synthesis of novel tetracycline derivatives with substitution at the C-8 position

✍ Scribed by Phaik-Eng Sum; Ving J. Lee; Francis P. Tally

Publisher: Elsevier Science
Year: 1994
Tongue: French
Weight: 148 KB
Volume: 35
Category: Article
ISSN: 0040-4039
DOI: 10.1016/s0040-4039(00)73173-x

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✦ Synopsis

I-Substituted te.mcycm. otiho&bmam' meS, ticatalyzed azide rearrangements. 7(or 9)-azimyclines Abstract llwC-8 funcdooalizatiooof te~clinederivatives via acid-catalyzed reatIangemf%It Of 7(or 9)azieyclines is c%zscribed. These ccmpomaaretbefifsttobepreparedfmulanin~ttehacyclincnucleus.

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