## Abstract A set of racemic spirocyclic quinuclidinyl‐Δ^2^‐isoxazoline derivatives was synthesized using a 1,3‐dipolar cycloaddition‐based approach. Target compounds were assayed for binding affinity toward rat neuronal homomeric (α7) and heteromeric (α4β2) nicotinic acetylcholine receptors. Δ^2^‐
✦ LIBER ✦
synthesis of new Δ2-isoxazoline derivatives and their pharmacological characterization as β-adrenergic receptor antagonists
✍ Scribed by Paola Conti; Clelia Dallanoce; Marco De Amici; Carlo De Micheli; Karl-Norbert Klotz
- Book ID
- 108480616
- Publisher
- Elsevier Science
- Year
- 1998
- Tongue
- English
- Weight
- 191 KB
- Volume
- 6
- Category
- Article
- ISSN
- 0968-0896
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