Chemistry of Aziridine Carboxylic Acids,
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Jähnisch, Klaus
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Article
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1997
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John Wiley and Sons
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English
⚖ 426 KB
## Abstract Enantiomerically pure __cis__‐ and __trans__‐1__H__‐aziridine‐carboxylic acid derivatives 2a, b and 3a, b have been prepared by asymmetric Michael‐type addition of ammonia to chiral acrylates 1a, b with high __syn__ selectivity. The title compounds were obtained from the diols 8a, b by