𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Synthesis of Indolines via a Domino Cu-Catalyzed Amidation/Cyclization Reaction

✍ Scribed by Minatti, Ana; Buchwald, Stephen L.

Book ID
115452003
Publisher
American Chemical Society
Year
2008
Tongue
English
Weight
134 KB
Volume
10
Category
Article
ISSN
1523-7060

No coin nor oath required. For personal study only.

πŸ“œ SIMILAR VOLUMES

Solid-phase synthesis of indolines via p
Solid-phase synthesis of indolines via palladium-catalyzed cyclization
✍ Yongping Yu; John M Ostresh; Richard A Houghten πŸ“‚ Article πŸ“… 2003 πŸ› Elsevier Science 🌐 French βš– 100 KB

The solid-phase synthesis of indolines from resin-bound 2-bromophenylacetylated amino acids is described. The exhaustive reduction of solid-support bound amides with borane afforded the requisite secondary amines that, following the palladium-catalyzed intramolecular cyclization and cleavage, provid