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Synthesis of high specific activity 17α-cyanomethyl-17β-hydroxy-[14α,15α-3H]estra-4,9-dien-3-one

✍ Scribed by P. Droescher; J. Röomer

Publisher
John Wiley and Sons
Year
1995
Tongue
French
Weight
377 KB
Volume
36
Category
Article
ISSN
0022-2135

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✦ Synopsis

Abstract

An improved synthesis of the tritium labelled form of the new pharmacon DIENOGEST is described. The [^14^α,15α‐^3^‐H]DIENOGEST was obtained with a specific activity of 51 Ci/mmol and a radiochemical purity > 98%.

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