## Abstract A new strategy toward the important class of benzomorphans is described. The key bond formation is based on an intramolecular Buchwald–Hartwig enolate arylation reaction. Thus, alkylation of piperidones with __ortho__‐bromobenzyl bromides provides the necessary substrates. In the presen
✦ LIBER ✦
Synthesis of Benzomorphan Analogues by Intramolecular Buchwald—Hartwig Cyclization.
✍ Scribed by Anton S. Khartulyari; Martin E. Maier
- Publisher
- John Wiley and Sons
- Year
- 2007
- Weight
- 19 KB
- Volume
- 38
- Category
- Article
- ISSN
- 0931-7597
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