𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Synthesis of an affinity ligand (‘UPHIT’) for in vivo acylation of the κ-opioid receptor

✍ Scribed by Brian R. de Costa; Linda Band; Richard B. Rothman; Arthur E. Jacobson; Victor Bykov; Agu Pert; Kenner C. Rice


Book ID
115921841
Publisher
Elsevier Science
Year
1989
Tongue
English
Weight
309 KB
Volume
249
Category
Article
ISSN
0014-5793

No coin nor oath required. For personal study only.


📜 SIMILAR VOLUMES


Synthesis of [3H]DIPPA: A potent irrever
✍ An-Chih Chang; Joseph D. Trometer; Philip S. Portoghese 📂 Article 📅 1995 🏛 John Wiley and Sons 🌐 French ⚖ 222 KB

## Abstract 2‐(3,4‐Dichlorophenyl)‐N‐methyl‐N‐[(1S)‐1‐(3‐isothiocyanatophenyl)‐2‐(1‐pyrrolidinyl)ethyl]acetamide (1, DIPPA) has been previously reported to be an opioid receptor affinity label that produces selective and long‐lasting κ opioid receptor antagonism in mice, High specific activity [^3^