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Synthesis of a phosphinic acid analogue of cyclic AMP

✍ Scribed by Andrew C. Regan; Nunzio Sciammetta; Peter I. Tattersall

Publisher
Elsevier Science
Year
2000
Tongue
French
Weight
101 KB
Volume
41
Category
Article
ISSN
0040-4039

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✦ Synopsis

Synthesis of a cyclic phosphinate ester analogue of cyclic AMP was achieved by using a double Arbuzov-type cyclisation of bis-trimethylsilyl phosphonite onto a sugar dihalide derivative as the key step.

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