Synthesis of 5-Acylindoles via Regioselective Acylation of 3-Trifluoroacetylindole.
β Scribed by Jun Li; Bogang Li; Xiaozhen Chen; Guolin Zhang
- Publisher
- John Wiley and Sons
- Year
- 2003
- Weight
- 107 KB
- Volume
- 34
- Category
- Article
- ISSN
- 0931-7597
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π SIMILAR VOLUMES
Reaction of 3-trifluoroacetylindole (4) with lithium dialkylamides affords the corresponding indole-3-carboxamides (5) in good to excellent yields.
## Abstract For Abstract see ChemInform Abstract in Full Text.
An efficient two-step synthesis of 8-acylated pyrazolo[1,5-a]-1,3,5-triazines has been accomplished. The key strategic elements of this novel synthetic approach involve the use of the N-methyl-N-phenylamino activating group, which was easily obtained in high yield by treatment of the pyrazolotriazin
## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 100 leading journals. To access a ChemInform Abstract of an article which was published elsewhere, please select a βFull Textβ option. The original article is trackable v