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Synthesis of (2S,1′ S,2′ S)-2-methyl-2-(carboxycyclopropyl)glycine and (S)-2-amino-2-methyl-4-phosphonobutyric acid from l-alanine

✍ Scribed by Dawei Ma; Zhaochun Ma; Jiqing Jiang; Zhen Yang; Chongzhi Zheng

Publisher
Elsevier Science
Year
1997
Tongue
English
Weight
324 KB
Volume
8
Category
Article
ISSN
0957-4166

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✦ Synopsis

The synthesis of two isotype-selective antagonists for metabotropic glutamate receptors, (2S, l'S,2'S)-2-methyl-2-(carboxycyclopropyl)glycine and (S)-2-amino-2methyl-4-phosphonobutyric acid from L-alanine is described. (~) 1997 Elsevier Science Ltd. All fights reserved.

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