Synthesis of 2-(5-Bromo-2,3-dimethoxyphenyl)-5-(aminomethyl)-1H-pyrrole analogues and their binding affinities for dopamine D2, D3, and D4 receptors
β Scribed by Robert H Mach; Yunsheng Huang; Rebekah A Freeman; Li Wu; Suwanna Blair; Robert R Luedtke
- Book ID
- 108479258
- Publisher
- Elsevier Science
- Year
- 2003
- Tongue
- English
- Weight
- 221 KB
- Volume
- 11
- Category
- Article
- ISSN
- 0968-0896
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Starting from 2-methyl-3-ethyl-lH-4,5,6,7-tetrahydroindol4one 3 we have prepared 2-methyl-3ethyl-5-morpholinoethyl-1H-4,5,6,7-tetmhydroindol4one. (1) and 2-methyl-3-ethyl-5-(4-o-methoxyphenyl-lpiperazinoethyl)-lH-4,5.6,7-tetrahydroindol-4-one (2) as butyrophenone analogues of the neuroleptic molindo