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Synthesis of 14C-labelled 1-β-D-arabinofuranosyl-E–5–(2-bromovinyl)uracil (BV-araU)

✍ Scribed by Masao Kumagai; Shinji Sakata; Toyofumi Yamaguchi; Kazuyoshi Ikeda; Haruhiko Machida

Publisher: John Wiley and Sons
Year: 1989
Tongue: French
Weight: 174 KB
Volume: 27
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.2580270503

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✦ Synopsis

1 4 C-Labelled l-~-D-arabinofuranosyl-E-5-(2-bromovinyl)uracil (BV-araU) was synthesized in 26.6% radiochemical yield from 1-R-Darabinofuranosyl-5-formyluracil and '"C-labelled malonic acid for the purpose of the metabolic studies in animals.

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