✦ LIBER ✦

Synthesis and Study of 5′-Ester Prodrugs of N6-Cyclopentyladenosine, a Selective A1 Receptor Agonist

✍ Scribed by Alessandro Dalpiaz; Angelo Scatturin; Enea Menegatti; Fabrizio Bortolotti; Barbara Pavan; Carla Biondi; Elisa Durini; Stefano Manfredini

Book ID: 110296667
Publisher: Springer US
Year: 2001
Tongue: English
Weight: 166 KB
Volume: 18
Category: Article
ISSN: 0724-8741
DOI: 10.1023/a:1011018730459

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Adenosine receptor prodrugs: Synthesis a

Adenosine receptor prodrugs: Synthesis and biological activity of derivatives of potent, A1-selective agonists

✍ Michel C. Maillard; Olga Nikodijević; Kathryn F. Lanoue; Deborah Berkich; Xiao-D 📂 Article 📅 1994 🏛 John Wiley and Sons 🌐 English ⚖ 977 KB

5'-Ester derivatives of the potent adenosine agonists N6-[4-[[[[4-[[[(2-acetylaminoethyl)amino]carbonyl]methyl] anilino]carbonyl]methyl]phenyl]adenosine (N-AcADAC; 1) and N6-cyclopentyladenosine (CPA; 2) were prepared as prodrugs. Both alkyl esters or carbonates (designed to enter the brain by virtu

The antinociceptive effect of 2-chloro-2

The antinociceptive effect of 2-chloro-2′-C-methyl-N6-cyclopentyladenosine (2′-Me-CCPA), a highly selective adenosine A1 receptor agonist, in the rat

✍ S. Maione; V. de Novellis; L. Cappellacci; E. Palazzo; D. Vita; L. Luongo; L. St 📂 Article 📅 2007 🏛 Elsevier Science 🌐 English ⚖ 740 KB

Interaction of the adenosine A1 receptor

Interaction of the adenosine A1 receptor agonist N6-cyclopentyladenosine (CPA) and opioid receptors in spinal cord nociceptive reflexes

✍ Ramos-Zepeda, Guillermo; Herrero, Juan F. 📂 Article 📅 2013 🏛 Elsevier Science 🌐 English ⚖ 938 KB

High-performance liquid chromatography o

High-performance liquid chromatography of the adenosine A1 agonist N6-cyclopentyladenosine and the A1 antagonist 8-cyclopentyltheophylline and its application in a pharmacokinetic study in rats

✍ R.A.A. Mathoˆt; S. Appel; E.A. van Schaick; W. Soudijn; A.P. Ijzerman; M. Danhof 📂 Article 📅 1993 🏛 Elsevier Science ⚖ 426 KB

Highly selective A1-adenosine-agonist (2

Highly selective A1-adenosine-agonist (2-chloro-N6-cyclopentyladenosine) and reduction of flap necrosis in adipocutaneous flaps in rats

✍ Andreas K. Dacho; Stefan Lyutenski; Gabriela Aust; Andreas Dietz 📂 Article 📅 2011 🏛 John Wiley and Sons 🌐 English ⚖ 313 KB

Synthesis and Biological Characterizatio

Synthesis and Biological Characterization of L-N 6 -(1-Iminoethyl)lysine 5-Tetrazole-amide, a Prodrug of a Selective iNOS Inhibitor

✍ Hallinan, E. Ann; Tsymbalov, Sofya; Dorn, Clifford R.; Pitzele, Barnett S.; Hans 📂 Article 📅 2002 🏛 American Chemical Society 🌐 English ⚖ 54 KB