✦ LIBER ✦

Synthesis and preliminary evaluation of [11C]KF15372, a selective adenosine A1 antagonist

✍ Scribed by Kiichi Ishiwata; Riko Furuta; Jun-Ichi Shimada; Shin-Ichi Ishii; Kazutoyo Endo; Fumio Suzuki; Michio Senda

Publisher: Elsevier Science
Year: 1995
Tongue: English
Weight: 405 KB
Volume: 46
Category: Article
ISSN: 0969-8043
DOI: 10.1016/0969-8043(95)00197-l

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis and preliminary evaluation of

Synthesis and preliminary evaluation of [11C]KF17837, a selective adenosine A2A antagonist

✍ Kiichi Ishiwata; Junko Noguchi; Hinako Toyama; Yojiro Sakiyama; Nobuaki Koike; S 📂 Article 📅 1996 🏛 Elsevier Science 🌐 English ⚖ 371 KB

An 11C-labeled selective adenosine A2A antagonist, (E)-8-(3,4-dimethoxystyryl)-1,3-dipropyl-7-[11C]-methylxanthine ([11C]KF17837), was prepared by reaction of (E)-8-(3,4-dimethoxystyryl)-1,3-dipropylxanthine and [11C]methyl iodide with decay-corrected radiochemical yield of 19-50%, radiochemical pur

Synthesis and evaluation of [11C]RU40555

Synthesis and evaluation of [11C]RU40555, a selective glucocorticoid receptor antagonist

✍ Takahiro Matsuya; Hiroyuki Takamatsu; Yoshihiro Murakami; Akihiro Noda; Kazuhiko 📂 Article 📅 2005 🏛 John Wiley and Sons 🌐 French ⚖ 224 KB

## Abstract We demonstrated the synthesis of carbon‐11 labeled 17‐__α__‐hydroxy‐11‐__β__‐/4‐/[methyl]‐[1‐methylethyl]‐aminophenyl/‐17__α__‐[prop‐1‐ynyl]esta‐4‐9‐diene‐3‐one (RU40555), a selective glucocorticoid receptor (GR) antagonist, and examined the __in vivo__ profile of [^11^C]RU40555. [^11^

ChemInform Abstract: Synthesis and Preli

ChemInform Abstract: Synthesis and Preliminary Evaluation of (S)-2-(4′-Carboxycubyl)glycine, a New Selective mGluR1 Antagonist.

✍ R. PELLICCIARI; G. COSTANTINO; E. GIOVAGNONI; L. MATTOLI; I. BRABET; J.-P. PIN 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 36 KB

Synthesis and in vivo evaluation of [11C

Synthesis and in vivo evaluation of [11C]semotiadil, a benzothiazine calcium antagonist

✍ Kiichi Ishiwata; Hiroyuki Seki; Kenji Ishii; Shin-Ichi Ishii; Tadashi Nozaki; Mi 📂 Article 📅 1994 🏛 Elsevier Science 🌐 English ⚖ 491 KB

Synthesis of an o-Nitrobenzyl Attached A

Synthesis of an o-Nitrobenzyl Attached A1 Adenosine Receptor Antagonist, a Prodrug Approach.

✍ HeXi Chang; Carol Ensinger; Robert D. McCargar; Bruno M. Vittimberga 📂 Article 📅 2003 🏛 John Wiley and Sons ⚖ 111 KB

## Abstract For Abstract see ChemInform Abstract in Full Text.

Synthesis and evaluation of 1,2,4-triazo

Synthesis and evaluation of 1,2,4-triazolo[1,5-c]pyrimidine derivatives as A2A receptor-selective antagonists

✍ Bidhan A. Shinkre; T. Santhosh Kumar; Zhan-Guo Gao; Francesca Deflorian; Kenneth 📂 Article 📅 2010 🏛 Elsevier Science 🌐 English ⚖ 645 KB

Movement disorders such as Parkinson's disease and Huntington's disease are serious life-limiting and debilitating movement disorders. Their onset typically occurs from mid-life to late in life, and effective diagnostic techniques for detecting and following the disease course are lacking. Our goal