The triflates and pivalates of 3 alpha-hydroxymethyl-6-substituted-2,2-dimethylpenam sulfones 3, 5; methyl and benzyl 6-substituted penicillanates 6-9 and 3-exo-methylene-6-substituted-2,2-dimethylpenam sulfone 4 were synthesized. These novel compounds were evaluated as elastase inhibitors using por
✦ LIBER ✦
Synthesis and porcine pancreatic elastase inhibitory evaluation of 6α-(sulfonyl)oxy-and 6α-chloropenicillanate sulfone esters and 3α-(acyloxy)methyl-6α-chloropenam sulfones
✍ Scribed by Carlos E. Boschetti; Ernesto G. Mata; Oreste A. Mascaretti; Julia A. Cricco; Gabriela Coux; Oscar A. Roveri
- Publisher
- Elsevier Science
- Year
- 1995
- Tongue
- English
- Weight
- 256 KB
- Volume
- 5
- Category
- Article
- ISSN
- 0960-894X
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