We have prepared (S)-5-chloro-3-[ 1251]iodo-2-methoxy-N-( l-azabicyclo[2.2.2]oct-3-yl)benzamide ([125I]DAIZAC, [ 1254-3) as a radioligand for characterization of the 5-HT-3 receptor. Preparation of the 3-tri-n-butylstannyl precursor was accomplished from the corresponding unlabeled DAIZAC by reactio
Synthesis and pharmacological characterization of [125I]MRS1898, a high-affinity, selective radioligand for the rat A3adenosine receptor
β Scribed by Zhan-Guo Gao; Bao Teng; Haitao Wu; Bhalchandra V. Joshi; Gary L. Griffiths; Kenneth A. Jacobson
- Publisher
- Springer Netherlands
- Year
- 2008
- Tongue
- English
- Weight
- 205 KB
- Volume
- 5
- Category
- Article
- ISSN
- 1573-9538
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