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Synthesis and evaluation of potent and selective human V1a receptor antagonists as potential ligands for PET or SPECT imaging

✍ Scribed by Karine Fabio; Christophe Guillon; Carl J. Lacey; Shi-fang Lu; Ned D. Heindel; Craig F. Ferris; Michael Placzek; Graham Jones; Michael J. Brownstein; Neal G. Simon

Book ID: 113495638
Publisher: Elsevier Science
Year: 2012
Tongue: English
Weight: 493 KB
Volume: 20
Category: Article
ISSN: 0968-0896
DOI: 10.1016/j.bmc.2011.12.013

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## Abstract We report the synthesis and evaluation of 1′‐(4‐[^125^I]iodobenzyl)‐3H‐spiro[isobenzofuran‐1,4′‐piperidine] ([^125^I]Spiro‐I) as a potential SPECT tracer for imaging of σ~1~ receptors. [^125^I]Spiro‐I was prepared in 55–65% isolated radiochemical yield, with radiochemical purity of >99%