A simple and efficient synthesis of a de
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Matthias Scheunemann; Bernd Johannsen
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Article
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1997
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Elsevier Science
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French
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A new approach to a pseudotripeptide based tetradentate chelating unit functionalizable with various bioactive groups has been developed. Using a one-pot reaction, a given 0)-aminoalkyl compound has been converted to a methylene thioether peptide isostere by two consecutive ring opening reactions.