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Synthesis and dopamine receptor affinity of (R)-(-)-2-fluoro-N-n-propylnorapomorphine: a highly potent and selective dopamine D2 agonist

✍ Scribed by Neumeyer, John L.; Gao, Yigong; Kula, Nora S.; Baldessarini, Ross J.

Book ID: 127207267
Publisher: American Chemical Society
Year: 1990
Tongue: English
Weight: 430 KB
Volume: 33
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm00174a002

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## Abstract 2‐Fluoronorapomorphine, the PET labelling precursor to 2‐fluoro‐__N__‐[^11^C]propylnorapomorphine, was prepared in 13 steps from codeine in a total yield of 10 %. Codeine was converted in four steps into __N__‐benzylnorcodeine which was oxidised by using the Swern protocol. Subsequent a