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Synthesis and configurational assignment of bicyclic “preactivated” analogues of cyclophosphamide

✍ Scribed by B. Lilo; M. Moreau; D. Bouchu

Publisher
Elsevier Science
Year
1990
Tongue
French
Weight
296 KB
Volume
31
Category
Article
ISSN
0040-4039

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✦ Synopsis

The synthesis of a new class of bicyclic "preactivated" analogues of Cyclophosphamide, 3-[bis(2-chloroethyl)MlinoJ-2-aza-3-phospha_4.10.4.O)&cane 3-oxide is described.

The configurational assignment of the stereoisomers was made by 31P and IH NMR.

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