✦ LIBER ✦

Synthesis and CNS Activity of Conformationally Restricted Butyrophenones. Part 27. New Synthetic Approaches to CNS Drugs. A Straightforward, Efficient Synthesis of Tetrahydroindol-4-ones and Tetrahydroquinolin-5-ones via Palladium-Catalyzed Oxidation of Hydroxyenaminones.

✍ Scribed by Beatriz Pita; Christian F. Masaguer; Enrique Ravina

Book ID: 101940803
Publisher: John Wiley and Sons
Year: 2003
Weight: 132 KB
Volume: 34
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.200304141

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✦ Synopsis

Abstract

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New synthetic approaches to CNS drugs. A

New synthetic approaches to CNS drugs. A straightforward, efficient synthesis of tetrahydroindol-4-ones and tetrahydroquinolin-5-ones via palladium-catalyzed oxidation of hydroxyenaminones

✍ Beatriz Pita; Christian F. Masaguer; Enrique Raviña 📂 Article 📅 2002 🏛 Elsevier Science 🌐 French ⚖ 97 KB

We have developed a facile and efficient synthesis of new conformationally restricted butyrophenones in the indole and quinoline series via palladium-catalyzed oxidation of hydroxyenaminones, and subsequent cyclization followed by spontaneous aromatization.