## Abstract A severe limitation in cancer therapy is the often insufficient differentiation between malign and benign tissue using known chemotherapeutics. One approach to decrease side effects is antibody‐directed enzyme prodrug therapy (ADEPT). We have developed new glycosidic prodrugs such as (−
✦ LIBER ✦
Synthesis and biological evaluations of a monomethylauristatin E glucuronide prodrug for selective cancer chemotherapy
✍ Scribed by Legigan, Thibaut; Clarhaut, Jonathan; Renoux, Brigitte; Tranoy-Opalinski, Isabelle; Monvoisin, Arnaud; Jayle, Christophe; Alsarraf, Jérôme; Thomas, Mikaël; Papot, Sébastien
- Book ID
- 123449989
- Publisher
- Elsevier Science
- Year
- 2013
- Tongue
- French
- Weight
- 547 KB
- Volume
- 67
- Category
- Article
- ISSN
- 0223-5234
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