✦ LIBER ✦

Synthesis and biological activity of NK1 tachykinin antagonists not containing D-residues

✍ Scribed by C. Poulos; M. Antoniou; R. Patacchini; C.A. Maggi; P. Rovero

Book ID: 113237341
Publisher: Elsevier Science
Year: 1994
Tongue: English
Weight: 255 KB
Volume: 26
Category: Article
ISSN: 0143-4179
DOI: 10.1016/0143-4179(94)90093-0

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis and biological activity of NK-

Synthesis and biological activity of NK-2 selective tachykinin antagonists containing D-tryptophan

✍ P. Rovero; V. Pestellini; R. Patacchini; S. Giuliani; C.A. Maggi; A. Meli; A. Gi 📂 Article 📅 1990 🏛 Elsevier Science 🌐 English ⚖ 156 KB

Design, Synthesis, and SAR of Tachykinin

Design, Synthesis, and SAR of Tachykinin Antagonists: Modulation of Balance in NK 1 /NK 2 Receptor Antagonist Activity

✍ Albert, Jeffrey S.; Aharony, David; Andisik, Donald; Barthlow, Herbert; Bernstei 📂 Article 📅 2002 🏛 American Chemical Society 🌐 English ⚖ 193 KB

ChemInform Abstract: Combined NK1 and NK

ChemInform Abstract: Combined NK1 and NK2 Tachykinin Receptor Antagonists: Synthesis and Structure—Activity Relationships of Novel Oxazolidine Analogues.

✍ Takahide Nishi; et al. et al. 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 36 KB 👁 2 views

Activity of peptide and non-peptide anta

Activity of peptide and non-peptide antagonists at peripheral NK-1 tachykinin receptors

✍ R. Patacchini; P. Santicioli; M. Astolfi; P. Rovero; G. Viti; C.A. Maggi 📂 Article 📅 1992 🏛 Elsevier Science 🌐 English ⚖ 135 KB

A review of the design, synthesis and bi

A review of the design, synthesis and biological activity of the bicyclic hexapeptide tachykinin NK2 antagonist MEN 10627

✍ Laura Quartara; Vincenzo Pavone; Carlo Pedone; Angelina Lombardi; Anna Rita Renz 📂 Article 📅 1996 🏛 Elsevier Science 🌐 English ⚖ 473 KB

Synthesis and biological activity of tac

Synthesis and biological activity of tachykinin analogs containing the adamantane moiety

✍ Daniela Pinzani; Anna Maria Papini; Mario Chelli; Mauro Ginanneschi; Carlo Alber 📂 Article 📅 1996 🏛 Springer Netherlands 🌐 English ⚖ 511 KB

2-adamantanole was the protecting group of the aspartate 13-COOH moiety during the peptide synthesis and survived the final peptide cleavage and deprotection carried out under controlled conditions. MEN 10586 showed an agonist activity comparable to that of the parent compound MEN 10210 at NK~ and N