2-Phenylquinolones as Inhibitors of the
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Barbara Gatto; Oriana Tabarrini; Serena Massari; Giulia Giaretta; Stefano Sabati
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Article
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2009
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John Wiley and Sons
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English
⚖ 202 KB
## Abstract **Novel 2‐phenylquinolones** aimed at the Tat–TAR complex were synthesized and tested. Derivatives characterized by precise modifications of the quinolone nucleus and to the side chain of the 2‐phenyl ring allowed a thorough structure–activity study, confirming 2‐phenylquinolone as a su