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Studies on pyrrolidinones. Synthesis of 1-[(N-acetylarylamino)methyl]pyroglutamic acid derivatives

✍ Scribed by Samira El Ghammarti; Benoit Rigo; Hechmi Mejdi; Jean-Pierre Hénichart; Daniel Couturier

Publisher
Journal of Heterocyclic Chemistry
Year
1998
Tongue
English
Weight
575 KB
Volume
35
Category
Article
ISSN
0022-152X

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✦ Synopsis

Abstract

Pyroglutamic acid was transformed into 1‐[(N‐Acetylarylamino)methyl]pyroglutamic acid derivatives by using trimethylsilyl variations of the Mannich reaction.

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