Conformation-activity relationships of c
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Sylwia Rodziewicz-MotowidŁo; Cezary Czaplewski; Sylwia Łuczak; Jerzy Ciarkowski
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Article
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2008
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John Wiley and Sons
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English
⚖ 233 KB
## Abstract The __N__‐terminal tetrapeptide segments of dermorphin (Tyr–D‐Ala–Phe–Gly–Tyr–Pro–Ser–NH~2~) and deltorphin (Tyr–D‐Ala–Phe–Asp/Glu–Val–Val–Gly–NH~2~) are agonists at the opioid receptors µ and δ, respectively. [D‐Arg^2^, Lys^4^]‐dermorphin‐(1–4) amide (Tyr–D‐Arg–Phe–Lys–NH~2~, DALDA) an