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Structure-activity relationship of bromoeudistomin D, a powerful Ca2+ releaser in skeletal muscle sarcoplasmic reticulum

✍ Scribed by Yukiko Takahashi; Ken-Ichi Furukawa; Masami Ishibashi; Daisuke Kozutsumi; Haruaki Ishiyama; Jun'ichi Kobayashi; Yasushi Ohizumi


Book ID
113398866
Publisher
Elsevier Science
Year
1995
Tongue
English
Weight
770 KB
Volume
288
Category
Article
ISSN
0922-4106

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Ca2+ release from skeletal sarcoplasmic reticulum (SR) could be regulated by at least three mechanisms: 1) Ca2+, 2) calmodulin, and 3) Ca2+/calmodulin-dependent phosphorylation. Bell-shaped Ca(2+)-dependence of Ca2+ release from both actively- and passively-loaded SR vesicles suggest that opening an