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Stereoselective synthesis of the C21C27 fragment of the phorboxazoles

✍ Scribed by Bo Liu; Wei-Shan Zhou

Publisher
Elsevier Science
Year
2003
Tongue
French
Weight
120 KB
Volume
44
Category
Article
ISSN
0040-4039

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✦ Synopsis

A stereoselective synthesis of the C21 C27 fragment of phorboxazoles A and B was achieved in 12 linear steps via an intramolecular cyclization induced by mercury acetate, to afford a functionalized tetrahydropyran.

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