A solid-phase synthesis of benzimidazoles, substituted on the aromatic ring by a variety of groups or atoms, is described. Intermediate 3, derived from the acylation of a resin-bound secondary amine with Fmoc-glycine, was elaborated via nucleophilic displacement with substituted o-halonitroarenes to
β¦ LIBER β¦
Solid phase synthesis of benzimidazoles
β Scribed by Gary B. Phillips; Guo Ping Wei
- Publisher
- Elsevier Science
- Year
- 1996
- Tongue
- French
- Weight
- 204 KB
- Volume
- 37
- Category
- Article
- ISSN
- 0040-4039
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