Solid-Phase Synthesis of 2-Amino-5-sulfa
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Marie Grimstrup; Florencio Zaragoza
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Article
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2002
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John Wiley and Sons
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English
⚖ 148 KB
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A solid-phase synthesis that provides easy access to 2-amino-5-sulfanylthiazoles with variable substituents at C-2, C-4, and C-5 has been developed. The key step of this synthesis is a new C-sulfanylation of resin-bound 2-aminothiazoles by mixtures of various sulfur-containing building blocks and io