𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Solid phase synthesis of 1,5-disubstituted pyrazole-4-hydroxamic acids and pyrazole-4-carboxamides via direct amidation of β-ketoesters

✍ Scribed by Weixu Zhai; Samuel W. Gerritz; Michael J. Sofia


Book ID
113930270
Publisher
Elsevier Science
Year
2012
Tongue
French
Weight
543 KB
Volume
53
Category
Article
ISSN
0040-4039

No coin nor oath required. For personal study only.


📜 SIMILAR VOLUMES


Solid-phase synthesis of 3,7-disubstitut
✍ Jérôme Giovannoni; Gilles Subra; Muriel Amblard; Jean Martinez 📂 Article 📅 2001 🏛 Elsevier Science 🌐 French ⚖ 71 KB

We report here the synthesis of 3,7-disubstituted perhydro-1,4-diazepine-2,5-diones from amino acids and b-amino acids using a backbone amide linker (BAL) as a cis-configuration inductor. We have optimized each steps of the synthesis on solid support using Mimotopes crowns.