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Selective reversible and irreversible ligands for the .kappa. opioid receptor

✍ Scribed by Cheng, Chen Yu; Wu, Shou Chien; Hsin, Ling Wei; Tam, S. William

Book ID: 120609855
Publisher: American Chemical Society
Year: 1992
Tongue: English
Weight: 753 KB
Volume: 35
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm00090a015

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## Abstract 2‐(3,4‐Dichlorophenyl)‐N‐methyl‐N‐[(1S)‐1‐(3‐isothiocyanatophenyl)‐2‐(1‐pyrrolidinyl)ethyl]acetamide (1, DIPPA) has been previously reported to be an opioid receptor affinity label that produces selective and long‐lasting κ opioid receptor antagonism in mice, High specific activity [^3^