A concise and efficient synthesis of highly enantioenriched 3-alkyl and 3-aryl-2,3-dihydro-1H-isoindolinones is reported. The key step relies on the diastereoselective reduction of the N-acylhydrazonium salts generated by acidic treatment of hemiaminal precursors bearing the (S)-2-methoxymethylpyrro
Rhodium complex-catalyzed desilylative cyclocarbonylation of 1-aryl-2-(trimethylsilyl)acetylenes: a new route to 2,3-dihydro-1H-inden-1-ones
✍ Scribed by Takeuchi, Ryo; Yasue, Hiroyuki
- Book ID
- 121419437
- Publisher
- American Chemical Society
- Year
- 1993
- Tongue
- English
- Weight
- 863 KB
- Volume
- 58
- Category
- Article
- ISSN
- 0022-3263
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