ChemInform Abstract: Regioselective N-Al
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G. BAR-HAIM; M. KOL
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Article
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2010
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John Wiley and Sons
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Regioselective N-Alkylation of 2-Aminobenzylamine via Chelation to 9-BBN. -Base-promoted alkylation of the easily available adduct (III) of 9-BBN and 2-aminobenzylamine results in high yield formation of a mono-substituted product (V). Final hydrolysis with HCl or NaOH leads to 2-amino-N-alkylbenzy