𝔖 Bobbio Scriptorium
✦   LIBER   ✦

Quantification of translocator protein (18 kDa) in the human brain with PET and a novel radioligand, [18F]-FEPPA

✍ Scribed by Pablo M. Rusjan; Alan A. Wilson; Peter M. Bloomfield; Sylvain Houle; Romina Mizrahi

Book ID
119331363
Publisher
Elsevier Science
Year
2010
Tongue
English
Weight
101 KB
Volume
52
Category
Article
ISSN
1053-8119

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Radiosynthesis of [18F]DPA-714, a select
Radiosynthesis of [18F]DPA-714, a selective radioligand for imaging the translocator protein (18 kDa) with PET
✍ Annelaure Damont; Françoise Hinnen; Bertrand Kuhnast; Marie-Anne Schöllhorn-Peyr 📂 Article 📅 2008 🏛 John Wiley and Sons 🌐 French ⚖ 193 KB

## Abstract Recently, a novel series of 2‐phenylpyrazolo[1,5‐__a__]pyrimidineacetamides has been reported as selective ligands of the translocator protein (18 kDa). Within this series, DPA‐714 (__N,N__‐diethyl‐2‐(2‐(4‐(2‐fluoroethoxy)phenyl)‐5,7‐dimethylpyrazolo[1,5‐__a__]pyrimidin‐3‐yl)acetamide,

Radiosynthesis of [18F]PBR111, a selecti
Radiosynthesis of [18F]PBR111, a selective radioligand for imaging the translocator protein (18 kDa) with PET
✍ Frédéric Dollé; Françoise Hinnen; Annelaure Damont; Bertrand Kuhnast; Christophe 📂 Article 📅 2008 🏛 John Wiley and Sons 🌐 French ⚖ 137 KB

## Abstract PBR111 (2‐(6‐chloro‐2‐(4‐(3‐fluoropropoxy)phenyl)imidazo[1,2‐__a__]pyridin‐3‐yl)‐__N__,__N__‐diethylacetamide) is a novel, reported, high‐affinity and selective ligand for the translocator protein (18 kDa). PBR111 has been labelled with fluorine‐18 (half‐life: 109.8 min) using our Zymat