𝔖 Bobbio Scriptorium
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Protease inhibitors and statins: pharmacokinetic interactions


Book ID
120863213
Publisher
Adis International Limited (now part of Wolters Kluwer Health)
Year
2002
Weight
139 KB
Volume
&NA;
Category
Article
ISSN
1173-8324

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✍ Hirokazu Yamaji; Yasuhiro Matsumura; Yukako Yoshikawa; Kanji Takada πŸ“‚ Article πŸ“… 1999 πŸ› John Wiley and Sons 🌐 English βš– 171 KB πŸ‘ 2 views

The interactions of four HIV-protease inhibitors, ritonavir (RIT), saquinavir (SAQ), indinavir (IND) and nelfinavir (NEL), were examined by in vitro metabolic studies using rat liver microsomal fractions. The substrate concentrations employed were 0.75 12 mM, and the inhibitor concentrations were 2.