Pharmacokinetic interactions between HIV
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Hirokazu Yamaji; Yasuhiro Matsumura; Yukako Yoshikawa; Kanji Takada
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Article
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1999
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John Wiley and Sons
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English
β 171 KB
π 2 views
The interactions of four HIV-protease inhibitors, ritonavir (RIT), saquinavir (SAQ), indinavir (IND) and nelfinavir (NEL), were examined by in vitro metabolic studies using rat liver microsomal fractions. The substrate concentrations employed were 0.75 12 mM, and the inhibitor concentrations were 2.