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Practical synthesis of α-aminoalkyl-α′-chloromethylketone derivatives. Part 1: Chloromethylation of N-protected 3-oxazolidin-5-ones

✍ Scribed by Tomoyuki Onishi; Naoko Hirose; Takashi Nakano; Masakazu Nakazawa; Kunisuke Izawa

Publisher
Elsevier Science
Year
2001
Tongue
French
Weight
69 KB
Volume
42
Category
Article
ISSN
0040-4039

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✦ Synopsis

Moc; Methoxycarbonyloxy group 3 1) TMSCl, n BuLi 2) BrCH 2 Cl, n BuLi 3 steps, 76%

  1. H +

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