✦ LIBER ✦

Piperazinyloxoquinoline derivatives, potent and selective inhibitors of HIV-1 transcription

✍ Scribed by M. Baba; M. Okamoto; M. Makini; Y. Kimura; T. Ikeuchi; T. Sakaguchi; T. Okamoto

Book ID: 114144961
Publisher: Elsevier Science
Year: 1997
Tongue: English
Weight: 105 KB
Volume: 34
Category: Article
ISSN: 0166-3542
DOI: 10.1016/s0166-3542(97)83146-4

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Mechanism of inhibition by piperazinylox

Mechanism of inhibition by piperazinyloxoquinoline derivatives as novel HIV-1 transcription inhibitors

✍ M. Okamoto; Y. Suruga; M. Makino; Y. Kimura; T. Ikeuchi; T. Sakaguchi; T. Okamot 📂 Article 📅 1997 🏛 Elsevier Science 🌐 English ⚖ 104 KB

Studies of Anti-HIV Transcription Inhibi

Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives

✍ Prof. Oriana Tabarrini; Dr. Serena Massari; Dr. Dirk Daelemans; Dr. Francesco Me 📂 Article 📅 2010 🏛 John Wiley and Sons 🌐 English ⚖ 416 KB 👁 1 views

## Abstract __The 6‐desfluoroquinolones (6‐DFQs) are anti‐HIV agents that target Tat‐mediated transcription. This particular mechanism of action makes this class of compounds very attractive for further structural investigations. Identification of the pharmacophore required for inhibition will ulti

Potent and selective inhibitors of gelat

Potent and selective inhibitors of gelatinase-a 1. hydroxamic acid derivatives

✍ John R. Porter; Nigel R.A. Beeley; Byron A. Boyce; Barbara Mason; Andrew Millica 📂 Article 📅 1994 🏛 Elsevier Science 🌐 English ⚖ 341 KB

Thiadiazole Derivatives: Highly Potent a

Thiadiazole Derivatives: Highly Potent and Specific HIV-1 Reverse Transcriptase Inhibitors

✍ Hanasaki, Yasuaki; Watanabe, Hiroyuki; Katsuura, Kimio; Takayama, Hiromitsu; Shi 📂 Article 📅 1995 🏛 American Chemical Society 🌐 English ⚖ 320 KB

Docking studies of flavonoid derivatives

Docking studies of flavonoid derivatives as potent HIV-1 integrase inhibitors

✍ Premjanu, N; Jaynthy, C; Soniyagandhi, C 📂 Article 📅 2014 🏛 BioMed Central 🌐 English ⚖ 86 KB

Inside Cover: Studies of Anti-HIV Transc

Inside Cover: Studies of Anti-HIV Transcription Inhibitor Quinolones: Identification of Potent N1-Vinyl Derivatives (ChemMedChem 11/2010)

✍ Prof. Oriana Tabarrini; Dr. Serena Massari; Dr. Dirk Daelemans; Dr. Francesco Me 📂 Article 📅 2010 🏛 John Wiley and Sons 🌐 English ⚖ 529 KB