✦ LIBER ✦

Peptidyl and azapeptidyl methylketones as substrate analog inhibitors of papain and cathepsin B

✍ Scribed by R Calabretta; C Giordano; C Gallina; V Morea; V Consalvi; R Scandurra

Book ID: 103630118
Publisher: Elsevier Science
Year: 1995
Tongue: French
Weight: 951 KB
Volume: 30
Category: Article
ISSN: 0223-5234
DOI: 10.1016/0223-5234(96)88312-7

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Analogy between active sites of cathepsi

Analogy between active sites of cathepsin B1 and papain

✍ H. Keilová; J. Turková 📂 Article 📅 1970 🏛 Elsevier Science 🌐 English ⚖ 108 KB

Peptidyl thioamides as substrates and in

Peptidyl thioamides as substrates and inhibitors of papain, and as probes of the kinetic significance of the oxyanion hole

✍ Foje, Kevin L.; Hanzlik, Robert P. 📂 Article 📅 1994 🏛 Elsevier Science 🌐 English ⚖ 583 KB

Irreversible inactivation of papain and

Irreversible inactivation of papain and cathepsin B by epoxidic substrate analogues

✍ C Giordano; C Gallina; V Consalvi; R Scandurra 📂 Article 📅 1990 🏛 Elsevier Science 🌐 French ⚖ 971 KB

Peptidyl aldehyde derivatives as potent

Peptidyl aldehyde derivatives as potent and selective inhibitors of cathepsin L

✍ Je-Tae Woo; Sanae Sigeizumi; Kohji Yamaguchi; Kikuo Sugimoto; Takeo Kobori; Tomo 📂 Article 📅 1995 🏛 Elsevier Science 🌐 English ⚖ 194 KB

Novel Peptidyl Aryl Vinyl Sulfones as Hi

Novel Peptidyl Aryl Vinyl Sulfones as Highly Potent and Selective Inhibitors of Cathepsins L and B

✍ Laura Mendieta; Anna Picó; Teresa Tarragó; Meritxell Teixidó; Marcos Castillo; L 📂 Article 📅 2010 🏛 John Wiley and Sons 🌐 English ⚖ 995 KB

## Abstract __Herein we present the design, synthesis, and evaluation of a structurally novel library of 20 peptidyl 3‐aryl vinyl sulfones as inhibitors of cathepsins L and B. The building blocks, described here for the first time, were synthesized in a highly efficient and enantioselective manner,

Substrate/propeptide-derived endo-epoxys

Substrate/propeptide-derived endo-epoxysuccinyl peptides as highly potent and selective cathepsin B inhibitors

✍ Norbert Schaschke; Irmgard Assfalg-Machleidt; Werner Machleidt; Luis Moroder 📂 Article 📅 1998 🏛 Elsevier Science 🌐 English ⚖ 77 KB