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Optimisation of 2-cyano-pyrimidine inhibitors of cathepsin K: Improving selectivity over hERG

✍ Scribed by Zoran Rankovic; Jiaqiang Cai; Jennifer Kerr; Xavier Fradera; John Robinson; Ashvin Mistry; William Finlay; George McGarry; Fiona Andrews; Wilson Caulfield; Iain Cumming; Maureen Dempster; John Waller; Wullie Arbuckle; Mark Anderson; Iain Martin; Ann Mitchell; Clive Long; Mark Baugh; Paul Westwood; Emma Kinghorn; Phil Jones; Joost C.M. Uitdehaag; Mario van Zeeland; Dominique Potin; Laurent Saniere; Andre Fouquet; François Chevallier; Hortense Deronzier; Cecile Dorleans; Eric Nicolai

Book ID: 104004822
Publisher: Elsevier Science
Year: 2010
Tongue: English
Weight: 967 KB
Volume: 20
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2010.08.101

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