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Novel two-step, one-pot synthesis of primary acylureas

✍ Scribed by Zili Xiao; Michael G. Yang; Andrew J. Tebben; Michael A. Galella; David S. Weinstein

Publisher: Elsevier Science
Year: 2010
Tongue: French
Weight: 247 KB
Volume: 51
Category: Article
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2010.09.003

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✦ Synopsis

A new procedure for the synthesis of primary acylureas from cyanamide and a variety of carboxylic acids is described. Under mild reaction conditions, the products were obtained in good yield from commercially available starting materials.

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