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Novel epoxysuccinyl peptides Selective inhibitors of cathepsin B, in vitro

✍ Scribed by Mitsuo Murata; Satsuki Miyashita; Chihiro Yokoo; Musaharu Tamai; Kazunori Hanada; Katsuo Hatayama; Takae Towatari; Takeshi Nikawa; Nobuhiko Katunuma

Book ID: 115924639
Publisher: Elsevier Science
Year: 1991
Tongue: English
Weight: 604 KB
Volume: 280
Category: Article
ISSN: 0014-5793
DOI: 10.1016/0014-5793(91)80318-w

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## Abstract __Herein we present the design, synthesis, and evaluation of a structurally novel library of 20 peptidyl 3‐aryl vinyl sulfones as inhibitors of cathepsins L and B. The building blocks, described here for the first time, were synthesized in a highly efficient and enantioselective manner,