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Nonsteroidal progesterone receptor ligands with unprecedented receptor selectivity

✍ Scribed by Stephen Palmer; Carolyn A Campen; George F Allan; Philip Rybczynski; Donna Haynes-Johnson; Amy Hutchins; Patricia Kraft; Margaret Kiddoe; Muh-Tsann Lai; Elizabeth Lombardi; Phyllis Pedersen; Gary Hodgen; Donald W Combs

Book ID: 117668073
Publisher: Elsevier Science
Year: 2000
Tongue: English
Weight: 172 KB
Volume: 75
Category: Article
ISSN: 0960-0760
DOI: 10.1016/s0960-0760(00)00134-5

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## Abstract Progesterone is one of the first nuclear receptor hormones to be described functionally and subsequently approached as a drug target. Because progesterone (**1**) affects both menstruation and gestation __via__ the progesterone receptor (PR), research aimed at modulating its activity is