New application of heterocyclic diazonium salts. Synthesis of pyrazolo[3,4-d][1,2,3]triazin-4-ones and imidazo[4,5-d][1,2,3]triazin-4-ones
β Scribed by Juan Pablo Colomer; Elizabeth Laura Moyano
- Publisher
- Elsevier Science
- Year
- 2011
- Tongue
- French
- Weight
- 603 KB
- Volume
- 52
- Category
- Article
- ISSN
- 0040-4039
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β¦ Synopsis
The pyrazolo [3,4-d][1,2,3]triazin-4-ones 3 and imidazo [4,5-d][1,2,3]triazin-4-ones 4 are analogs structurally related to purines that have showed a wide and significant variety of biological activity. These compounds were synthesized by one-pot diazotization of 5-amino-1H-pyrazole-4-carbonitriles 1 and 5-amino-1H-imidazole-4-carbonitriles 2, respectively.
π SIMILAR VOLUMES
## Abstract Some novel 3,7βdimethylβ6__H__βpyrazolo[5,1βc][1,2,4]triazinβ4βones were prepared **(3aβg)**. Compounds **3a,b** were treated with hydrazines to afford various products **7a,b, 8a,b, 9 and lla,b** depending on the type of hydrazine derivative and reaction conditions. The benzoyloxyimino