✦ LIBER ✦

N-hydroxysulfamides as analog of N-hydroxyurea: synthesis and biological evaluation

✍ Scribed by A.-Houssem Hajri; Georges Dewynter; Marc Criton; Pierre Dilda; Jean-Louis Montero

Publisher: John Wiley and Sons
Year: 2001
Tongue: English
Weight: 82 KB
Volume: 12
Category: Article
ISSN: 1042-7163
DOI: 10.1002/1098-1071(2001)12:1<1::aid-hc1>3.0.co;2-q

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✦ Synopsis

A series of sulfa-analog of hydroxyurea, derived from N-hydroxysulfamide H 2 NSO 2 NHOH, were synthesized starting from chlorosulfonyl isocyanate (CSI) and O-substituted hydroxylamines. Their antiproliferative, antiviral (in synergy with ddI), and antifungal activities have been evaluated.

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