## Abstract Cycloaddition of the azide derivative **5** with 1,4‐dihydroxybutyne afforded the __N__‐thio‐acyclic nucleoside **6**, which prepared alternatively from coupling of the bromo derivative **8** with 2‐acetoxy‐ethylmercaptan. Deblocking of **6** gave the free nucleoside **7**. Mesylation o
N- and C-Acyclic Thionucleoside Analogues of 1,2,3-Triazole.
✍ Scribed by Najim A. Al-Masoudi; Yaseen A. Al-Soud; Asmehan Abdul-Zahra
- Publisher
- John Wiley and Sons
- Year
- 2004
- Weight
- 25 KB
- Volume
- 35
- Category
- Article
- ISSN
- 0931-7597
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