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N -[6-Amino-2-(heteroaryl)pyrimidin-4-yl]acetamides as A 2A Receptor Antagonists with Improved Drug Like Properties and in Vivo Efficacy

✍ Scribed by Lanier, Marion C.; Moorjani, Manisha; Luo, Zhiyong; Chen, Yongsheng; Lin, Emily; Tellew, John E.; Zhang, Xiaohu; Williams, John P.; Gross, Raymond S.; Lechner, Sandra M.; Markison, Stacy; Joswig, Tanya; Kargo, William; Piercey, Jaime; Santos, Mark; Malany, Siobhan; Zhao, Marilyn; Petroski, Robert; Crespo, María I.; Díaz, José-Luis; Saunders, John; Wen, Jenny; O’Brien, Zhihong; Jalali, Kayvon; Madan, Ajay; Slee, Deborah H.

Book ID: 120317591
Publisher: American Chemical Society
Year: 2009
Tongue: English
Weight: 461 KB
Volume: 52
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm800908d

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