Conformational searches on three closely related pp60 c-src protein tyrosine kinase inhibitors of varying potencies were performed to determine a structural basis for their activity. The first was a linear peptide (PDNEYAFFQf), the second its 10-membered cyclic analogue, and the third a cyclic analo
Measurement of the Protein Tyrosine Kinase Activity of c-src Using Time-Resolved Fluorometry of Europium Chelates
β Scribed by Albert F. Braunwalder; Donna R. Yarwood; Matthew A. Sills; Kenneth E. Lipson
- Publisher
- Elsevier Science
- Year
- 1996
- Tongue
- English
- Weight
- 102 KB
- Volume
- 238
- Category
- Article
- ISSN
- 0003-2697
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