✦ LIBER ✦

Interaction of linear and cyclic peptide antagonists at the human B2 kinin receptor

✍ Scribed by Paola Cucchi; Stefania Meini; Laura Quartara; Alessandro Giolitti; Sabrina Zappitelli; Luigi Rotondaro; Carlo Alberto Maggi

Book ID: 117408353
Publisher: Elsevier Science
Year: 2002
Tongue: English
Weight: 104 KB
Volume: 23
Category: Article
ISSN: 0196-9781
DOI: 10.1016/s0196-9781(02)00081-5

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

New conformationally homogeneous β-turn

New conformationally homogeneous β-turn antagonists of the human B2 kinin receptor

✍ Edith S. Monteagudo; Federico Calvani; Fernando Catrambone; Christopher I. Finch 📂 Article 📅 2001 🏛 John Wiley and Sons 🌐 English ⚖ 241 KB

## Abstract We have designed and synthesized a conformationally homogeneous series of cyclic pentapeptides of the general structure __c__[Pro‐aa~__i__~‐𝒹‐Tic‐Oic‐aa~__i__+3~] which adopt a type‐II′ β‐turn conformation believed important for high affinity antagonism of the bradykinin (BK) B~2~ recep

Solid-phase synthesis of MEN 11270, a ne

Solid-phase synthesis of MEN 11270, a new cyclic peptide kinin B2 receptor antagonist

✍ Beatrice Anichini; Renzo Ricci; Gaetano Fabbri; Giuseppe Balacco; Sandro Mauro; 📂 Article 📅 2000 🏛 John Wiley and Sons 🌐 English ⚖ 159 KB

The actions of kinin antagonists on B1 a

The actions of kinin antagonists on B1 and B2 receptor systems

✍ Domenico Regoli; Guy Drapeau; Paolo Rovero; Stéphane Dion; Pedro D'Orléans-Juste 📂 Article 📅 1986 🏛 Elsevier Science 🌐 English ⚖ 352 KB

Effects of two novel non-peptide antagon

Effects of two novel non-peptide antagonists at the rabbit bradykinin B2 receptor

✍ François Marceau; Steeve Houle; Johanne Bouthillier; Najeeb B. Said; Peter J. Ga 📂 Article 📅 2001 🏛 Elsevier Science 🌐 English ⚖ 274 KB

Site-directed mutagenesis at the human B

Site-directed mutagenesis at the human B2 receptor and molecular modelling to define the pharmacophore of non-peptide bradykinin receptor antagonists

✍ Stefania Meini; Paola Cucchi; Francesca Bellucci; Claudio Catalani; Angela Faiel 📂 Article 📅 2004 🏛 Elsevier Science 🌐 English ⚖ 277 KB

The use of kinin B1 and B2 receptor knoc

The use of kinin B1 and B2 receptor knockout mice and selective antagonists to characterize the nociceptive responses caused by kinins at the spinal level

✍ Juliano Ferreira; Maria M Campos; Ronaldo Araújo; Michael Bader; João B Pesquero 📂 Article 📅 2002 🏛 Elsevier Science 🌐 English ⚖ 162 KB