✦ LIBER ✦

Inhibitors of protein tyrosine kinases

✍ Scribed by David W Fry; Alexander J Bridges

Publisher: Elsevier Science
Year: 1995
Tongue: English
Weight: 745 KB
Volume: 6
Category: Article
ISSN: 0958-1669
DOI: 10.1016/0958-1669(95)80109-x

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✦ Synopsis

The description in the past year of several novel protein tyrosine kinase inhibitors, which exhibit dramatic improvements in potency and specificity over earlier agents, will be considered a major turning point in the field. These compounds appear to have the necessary pharmacological properties to finally allow clarification of whether suppression of specific tyrosine kinases is of therapeutic benefit in certain disease states.

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